SCHEMBL16113759

SCHEMBL16113759

CCCCOC(=O)Nc1ncc(C(=O)OCC)o1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.48
RAB9A P51151 9/20 0.48
NPC1 O15118 8/20 0.48
SMN1; SMN2 Q16637 8/20 0.48
TSHR P16473 4/20 0.48
CYP1A2 P05177 4/20 0.48
CYP2C19 P33261 4/20 0.48
HPGD P15428 4/20 0.48
CYP2C9 P11712 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.46
CASP1 P29466 1/20 0.44
MAPK1 P28482 2/20 0.43
CSNK2A2 P19784 1/20 0.42
CSNK2A1 P68400 1/20 0.42
ALDH1A1 P00352 3/20 0.42
HSD17B10 Q99714 1/20 0.42
NFKB1 P19838 1/20 0.42
STAT1 P42224 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12491653 0.81 NLRP3 (0.49) NLRP3TSHRALDH1A1KDM4EMAPT
SCHEMBL12852006 0.78 NLRP3 (0.56) NLRP3RAB9ANPC1SMN1; SMN2TSHR
SCHEMBL20267305 0.76 TSHR (0.46) SMN1; SMN2TSHRCYP1A2CYP2C19CYP2C9
SCHEMBL31716404 0.72 NLRP3 (0.43) NLRP3RAB9ANPC1SMN1; SMN2TSHR
SCHEMBL12481786 0.72 TSHR (0.60) RAB9ANPC1SMN1; SMN2TSHRCYP1A2
SCHEMBL28433114 0.71 HDAC4 (0.59) RAB9ANPC1SMN1; SMN2TSHRCYP1A2
SCHEMBL23812921 0.71 NLRP3 (0.56) NLRP3RAB9ANPC1MAPK1ALDH1A1
SCHEMBL3992206 0.71 NLRP3 (0.56) NLRP3RAB9ANPC1SMN1; SMN2HPGD
SCHEMBL3715054 0.71 NLRP3 (0.48) NLRP3RAB9ANPC1TSHRCYP1A2
SCHEMBL23731345 0.70 NLRP3 (0.52) NLRP3RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970272-A1 GLYCOSIDASE INHIBITORS Merck Patent GmbH (DE) 2016-01-20 EP disclosed
WO-2014159234-A1 GLYCOSIDASE INHIBITORS MERCK PATENT GMBH (DE) 2014-10-02 WO disclosed