SCHEMBL16116222

SCHEMBL16116222

COC(=O)c1cc(-c2ccnc(NC(=O)OC(C)(C)C)c2)c[nH]1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 2/20 0.45
ATR Q13535 1/20 0.45
AAK1 Q2M2I8 10/20 0.43
CCNC P24863 3/20 0.43
CDK8 P49336 3/20 0.43
IRAK4 Q9NWZ3 1/20 0.42
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41
TGFBR1 P36897 1/20 0.40
CYP3A4 P08684 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16115220 0.90 CCNC (0.43) PIK3C3ATRAAK1CCNCCDK8
SCHEMBL5548970 0.81 ATR (0.48) PIK3C3ATRAAK1IRAK4GSK3B
SCHEMBL16116380 0.78 CCNC (0.68) CCNCCDK8CYP3A4ALDH1A1LMNA
SCHEMBL5251219 0.78 EGFR (0.57) PIK3C3AAK1IRAK4GSK3BDYRK1A
SCHEMBL12127932 0.77 FDPS (0.54) PIK3C3AAK1GSK3BDYRK1AALDH1A1
SCHEMBL29992322 0.77 AAK1 (0.48) PIK3C3AAK1IRAK4GSK3BDYRK1A
SCHEMBL8670718 0.77 FDPS (0.50) PIK3C3AAK1IRAK4GSK3BDYRK1A
SCHEMBL17643492 0.77 AAK1 (0.48) PIK3C3AAK1IRAK4GSK3BDYRK1A
SCHEMBL16115068 0.76 CCNC (0.70) CCNCCDK8DYRK1AALDH1A1LMNA
SCHEMBL16116358 0.76 CCNC (0.51) CCNCCDK8ALDH1A1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014154723-A1 NOVEL PYRROLE DERIVATIVES FOR THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2014-10-02 WO disclosed
WO-2014154723-A1 NOVEL PYRROLE DERIVATIVES FOR THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2014-10-02 WO disclosed