SCHEMBL161180

SCHEMBL161180

COc1cc(C(=O)NN)ccc1-c1ccnc(C)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 2/20 0.48
PSEN2 P49810 2/20 0.48
APH1B Q8WW43 2/20 0.48
NCSTN Q92542 2/20 0.48
APH1A Q96BI3 2/20 0.48
PSENEN Q9NZ42 2/20 0.48
MKNK1 Q9BUB5 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46
ROCK2 O75116 4/20 0.45
ROCK1 Q13464 4/20 0.45
HDAC8 Q9BY41 1/20 0.45
WNT3A P56704 2/20 0.44
NOX1 Q9Y5S8 1/20 0.44
AAK1 Q2M2I8 2/20 0.44
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
PKM P14618 1/20 0.43
KMT2A Q03164 1/20 0.43
SCN9A Q15858 1/20 0.43
PTAFR P25105 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL155440 0.99 PSEN1 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL30637340 0.76 KDM4E (0.55) ALDH1A1
SCHEMBL1543956 0.76 KDM4E (0.55) ALDH1A1
SCHEMBL12302693 0.76 WNT3A (0.53) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2183834 0.76 PSEN1 (0.58) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2183830 0.76 WNT3A (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL29637091 0.76 DYRK1A (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1492639 0.76 DYRK1A (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL12516813 0.75 DYRK1A (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL18115543 0.75 USP30 (0.75)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611805-A1 FUSED TRIAZOLES FOR THE TREATMENT OR PROPHYLAXIS OF MILD COGNITIVE IMPAIRMENT Takeda Pharmaceutical Company Limited (JP) 2013-07-10 EP disclosed
WO-2012029991-A1 FUSED TRIAZOLES FOR THE TREATMENT OR PROPHYLAXIS OF MILD COGNITIVE IMPAIRMENT TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-08 WO disclosed