SCHEMBL16129753

SCHEMBL16129753

O=C(OCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)N1CCn2nc(C(=O)N3CCNCC3)cc2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 6/20 0.39
SCN7A Q01118 4/20 0.39
KCNH2 Q12809 3/20 0.39
ENPP2 Q13822 5/20 0.38
ATXN2 Q99700 3/20 0.38
HTR2A P28223 1/20 0.38
ABAT P80404 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
TACR1 P25103 5/20 0.37
CYP2D6 P10635 2/20 0.36
CYP3A4 P08684 1/20 0.36
CACNA1H O95180 1/20 0.36
USP2 O75604 1/20 0.36
SCN5A Q14524 1/20 0.36
SCN2A Q99250 1/20 0.36
SCN8A Q9UQD0 1/20 0.36
SCN10A Q9Y5Y9 1/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16093743 0.94 SCN9A (0.38) SCN9ASCN7AKCNH2ENPP2ATXN2
SCHEMBL16129902 0.94 ENPP2 (0.46) SCN9ASCN7AKCNH2ENPP2ATXN2
SCHEMBL16129760 0.91 TACR1 (0.38) ENPP2ATXN2HTR2AABATSIGMAR1
SCHEMBL16129885 0.90 TACR1 (0.38) ENPP2ATXN2HTR2AABATSIGMAR1
SCHEMBL16129893 0.90 TACR1 (0.39) SCN9AENPP2ATXN2HTR2AABAT
SCHEMBL16129767 0.89 SCN9A (0.41) SCN9AKCNH2ENPP2ATXN2HTR2A
SCHEMBL16129852 0.89 ENPP2 (0.45) SCN9ASCN7AKCNH2ENPP2ATXN2
SCHEMBL16129746 0.89 ENPP2 (0.37) ENPP2ATXN2HTR2AABATSIGMAR1
SCHEMBL16129897 0.88 TACR1 (0.47) ENPP2ATXN2TACR1CYP2D6CYP3A4
SCHEMBL16129896 0.88 ENPP2 (0.37) SCN9AENPP2ATXN2HTR2AABAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014152725-A1 S1P AND/OR ATX MODULATING AGENTS BIOGEN IDEC MA INC. (US) 2014-09-25 WO disclosed