SCHEMBL16153176

SCHEMBL16153176

C/N=C(/C)NC(=O)c1cc2cc(-c3cc(C(=O)NCc4ccc(C(=O)O)cc4)ncc3C)ccc2[nH]1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 4/20 0.59
AURKA O14965 1/20 0.50
MMP2 P08253 1/20 0.50
MMP10 P09238 1/20 0.50
MMP9 P14780 1/20 0.50
PRKACA P17612 1/20 0.50
DRD5 P21918 1/20 0.50
MAPKAPK2 P49137 1/20 0.50
MMP14 P50281 1/20 0.50
PRKAA1 Q13131 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1314036 0.78 MMP13 (0.55) MMP13
SCHEMBL1316043 0.74 MMP13 (1.00) MMP13AURKAMMP2MMP10MMP9
SCHEMBL1316395 0.72 MMP13 (0.73) MMP13AURKAMMP2MMP10MMP9
SCHEMBL1313634 0.69 MMP13 (1.00) MMP13AURKAMMP2MMP10MMP9
SCHEMBL15888040 0.69 MMP13 (0.54) MMP13MMP2MMP14
SCHEMBL1313851 0.68 MMP13 (0.68) MMP13
Bi 4394 SCHEMBL1314835 0.67 MMP13 (1.00) MMP13AURKAMMP2MMP10MMP9
SCHEMBL1313998 0.66 MMP13 (0.59) MMP13AURKAMMP2MMP10MMP9
SCHEMBL28954653 0.66 NAMPT (0.78)
SCHEMBL1316251 0.66 MMP13 (0.60) MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2340243-B1 HETEROARYL SUBSTITUTED INDOLE COMPOUNDS USEFUL AS MMP-13 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2014-10-08 EP disclosed