SCHEMBL16158487

SCHEMBL16158487

Nc1ccc2cc(-c3cccc(-n4cnc5ccccc54)c3)ccc2c1

nearest known ligand 0.68

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 7/20 0.55
HTT P42858 4/20 0.51
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
PTK2B Q14289 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
KDR P35968 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16158486 0.89 FGFR1 (0.59) FGFR1HTTKDM4EALDH1A1RAB9A
SCHEMBL2642019 0.88 FGFR1 (0.60) FGFR1HTTKDM4EALDH1A1RAB9A
SCHEMBL16147532 0.85 FGFR1 (0.68) FGFR1HTTMAPTKMT2APTK2B
SCHEMBL16147183 0.82 FGFR1 (0.74) FGFR1HTTALDH1A1KDR
SCHEMBL22329065 0.82 FGFR1 (0.53) FGFR1HTTKDM4EALDH1A1RAB9A
SCHEMBL4015486 0.82 HTT (0.71) FGFR1HTTMAPTKMT2APTK2B
SCHEMBL2306019 0.82 FGFR1 (0.67) FGFR1HTTKDM4EALDH1A1RAB9A
SCHEMBL16148290 0.81 FGFR1 (0.64) FGFR1HTTALDH1A1KDR
SCHEMBL16147687 0.81 FGFR1 (0.51) FGFR1HTTKDM4EALDH1A1RAB9A
SCHEMBL2643550 0.81 FGFR1 (0.78) FGFR1HTTALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014165815-A2 NONSTEROIDAL AND STEROIDAL COMPOUNDS WITH POTENT ANDROGEN RECEPTOR DOWN-REGULATION AND ANTI PROSTATE CANCER ACTIVITY UNIVERSITY OF MARYLAND, BALTIMORE (US) 2014-10-09 WO disclosed