SCHEMBL16162016

SCHEMBL16162016

CNCC(Nc1ncnc2c(OC(N)=O)cccc12)c1cccc(NC(=O)c2ccc(Br)cc2)c1

nearest known ligand 0.79

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AURKA O14965 20/20 0.79
RPS6KB1 P23443 19/20 0.79
AURKB Q96GD4 5/20 0.64
PDPK1 O15530 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16162095 0.93 AURKA (0.79) AURKARPS6KB1AURKBPDPK1
SCHEMBL16162101 0.91 AURKA (0.81) AURKARPS6KB1AURKBPDPK1
SCHEMBL16161955 0.91 AURKA (0.68) AURKARPS6KB1AURKBPDPK1
SCHEMBL16162051 0.91 AURKA (0.80) AURKARPS6KB1AURKB
SCHEMBL16162091 0.89 AURKA (0.81) AURKARPS6KB1AURKB
SCHEMBL16162121 0.89 AURKA (0.80) AURKARPS6KB1AURKB
SCHEMBL667172 0.89 AURKA (1.00) AURKARPS6KB1AURKBPDPK1
SCHEMBL16162135 0.88 AURKA (0.71) AURKARPS6KB1AURKBPDPK1
SCHEMBL16162061 0.87 AURKA (0.84) AURKARPS6KB1AURKB
SCHEMBL16161952 0.86 RPS6KB1 (0.79) AURKARPS6KB1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396307-B1 NOVEL AMINO AZAHETEROCYCLIC CARBOXAMIDES MERCK PATENT GMBH (DE) 2014-10-15 EP claimed