Thiophene

Thiophene

SCHEMBL1616682

O=C(O)O.c1ccsc1

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Thiophene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Thiophene SCHEMBL20482064 1.00 CA1 (0.39)
Oxalic Acid SCHEMBL6961961 0.89 DAO (0.32)
Oxalic Acid SCHEMBL28318799 0.89 DAO (0.32)
Thiophene SCHEMBL28550995 0.86 LCK (0.47)
Oxalic Acid SCHEMBL7447158 0.86 DAO (0.31)
Acetic Acid SCHEMBL29616843 0.86 LCK (0.47)
Oxalic Acid SCHEMBL7447155 0.86 DAO (0.31)
Oxalic Acid SCHEMBL6967440 0.86 DAO (0.31)
Thiophene SCHEMBL502436 0.86
Acetic Acid SCHEMBL755556 0.86 LCK (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150251158-A1 Functionalized Particulate Support Material and Methods of Making and Using the Same W. R. GRACE & CO.-CONN. (US) 2015-09-10 US claimed
EP-2811983-A1 FUNCTIONALIZED PARTICULATE SUPPORT MATERIAL AND METHODS OF MAKING AND USING THE SAME W.R. Grace & CO. - CONN. (US) 2014-12-17 EP claimed
WO-2014043644-A1 FUNCTIONALIZED PARTICULATE SUPPORT MATERIAL AND METHODS OF MAKING AND USING THE SAME ALLTECH ASSOCIATES, INC. (US) 2014-03-20 WO claimed
CN-115058743-B Novel composite electrolyte and method for refining secondary aluminum by low-temperature electrolysis 昆明理工大学 2024-05-24 CN disclosed
US-11529610-B2 Functionalized particulate support material and methods of making and using the same W.R. GRACE & CO.-CONN. (US) 2022-12-20 US disclosed
CN-113574059-A Modified ionic liquids containing a cyclic phosphorus moiety 诺姆斯科技股份有限公司 2021-10-29 CN disclosed
US-10717866-B2 Organic-inorganic hybrid composition, and article and optical component including the same SAMSUNG ELECTRONICS CO., LTD. (KR) 2020-07-21 US disclosed
EP-2811983-B1 FUNCTIONALIZED PARTICULATE SUPPORT MATERIAL AND METHODS OF MAKING AND USING THE SAME GRACE W R & CO (US) 2019-05-01 EP disclosed
US-20180244915-A1 ORGANIC-INORGANIC HYBRID COMPOSITION, AND ARTICLE AND OPTICAL COMPONENT INCLUDING THE SAME SAMSUNG ELECTRONICS CO., LTD. (KR) 2018-08-30 US disclosed
CN-103118651-B For microencapsulation compositions and the method for tissue mineralization PREMIER DENTAL PRODUCTS COMPNAY (US) 2016-01-06 CN disclosed
US-20150251158-A1 Functionalized Particulate Support Material and Methods of Making and Using the Same W. R. GRACE & CO.-CONN. (US) 2015-09-10 US disclosed
US-6555699-B2 Antitumor and antirheumatic agents, high binding affinity CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-04-29 US disclosed
US-20020193616-A1 16-ENE-VITAMIN D DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-12-19 US disclosed
US-6433200-B1 ANTITUMOR AND ANTIRHEUMATIC AGENTS, HIGH BINDING AFINITY TO VITAMIN D RECEPTORS AND WEAK HYPERCALCEMIC ACTIVITY CHUGEI SEIYAKU KABUSHIKI KAISHA (JP) 2002-08-13 US disclosed
US-20020032340-A1 16-ene-vitamin D derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-03-14 US disclosed
US-6326503-B1 ANTITUMOR AGENTS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-12-04 US disclosed
US-6184398-B1 ANTITUMOR AGENTS AND TREATMENT OF RHEUMATIC CONDITIONS; HIGH BINDING ABILITY TO VITAMIN D RECEPTORS AND WEAK HYPERCALCEMIC ACTIVITY; E.G.,1,3-DIHYDROXY-20-3-HYDROXY-3-METHYLBUTYLTHIO)-9,10-SECOPREGNA -5,7,10(19),16-TETRAENE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-02-06 US disclosed
EP-0947504-A1 16-ENE-VITAMIN D DERIVATIVES Chugai Seiyaku Kabushiki Kaisha (JP) 1999-10-06 EP disclosed
EP-0353753-A1 Amide compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1990-02-07 EP disclosed
US-4036972-A 2-(N-thienylmethyl-phenylamino)-imidazolines-(2) and salts thereof BOEHRINGER INGELHEIM GMBH (DT) 1977-07-19 US disclosed