SCHEMBL16169019

SCHEMBL16169019

C[C@@H](COS(C)(=O)=O)Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TAAR1 Q96RJ0 5/20 0.42
SLC6A2 P23975 3/20 0.42
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
SIGMAR1 Q99720 2/20 0.42
MAOA P21397 1/20 0.42
CYP2A6 P11509 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
TSHR P16473 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
HTR2A P28223 1/20 0.41
ADRA1A P35348 1/20 0.41
OPRK1 P41145 1/20 0.41
KCNH2 Q12809 1/20 0.41
SLC18A2 Q05940 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14388004 1.00 NPC1 (0.43) NPC1RAB9ATAAR1SLC6A2SLC6A4
SCHEMBL18063430 0.84 CA1 (0.57) TAAR1SLC6A2SLC6A4SLC6A3SIGMAR1
SCHEMBL4756135 0.84 CA1 (0.40) TAAR1SLC6A2SLC6A4SLC6A3SIGMAR1
SCHEMBL4756128 0.84 CA1 (0.40) TAAR1SLC6A2SLC6A4SLC6A3SIGMAR1
SCHEMBL9276273 0.81 TSHR (0.44) NPC1RAB9ATSHRMEN1KMT2A
SCHEMBL10501340 0.81 HTR2A (0.51) SIGMAR1CYP2A6HTR2A
SCHEMBL6953092 0.81 EPHX1 (0.53) TAAR1SLC6A2SLC6A4SLC6A3SIGMAR1
SCHEMBL11044498 0.81 TSHR (0.40) TAAR1SLC6A2SLC6A4SLC6A3SIGMAR1
SCHEMBL17443109 0.80 MCHR1 (0.44) TSHRMEN1KMT2A
SCHEMBL11045387 0.79 MEN1 (0.38) TAAR1SLC6A2SLC6A4SLC6A3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9051310-B2 Nicotinamide derivative or salt thereof FUJIFILM CORPORATION (JP) 2015-06-09 US disclosed
US-20140309225-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2014-10-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140309225-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF SYK, BTK, NOX4 NPC1 1823/4885RAB9A 2530/4885TAAR1 1991/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.