SCHEMBL16195686

SCHEMBL16195686

NC1(NO)CC(=O)NC1=O

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CYP19A1 P11511 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637001 0.69
SCHEMBL4356813 0.64 CYP19A1 (0.36) TSHRNPSR1CYP19A1
SCHEMBL1322984 0.64 CYP19A1 (0.36) TSHRNPSR1CYP19A1
SCHEMBL1325877 0.64 CYP19A1 (0.36) TSHRNPSR1CYP19A1
SCHEMBL10028354 0.64
SCHEMBL10025159 0.64
SCHEMBL3255645 0.62
SCHEMBL13805603 0.61 TSHR (0.44) TSHRNPSR1CYP19A1
SCHEMBL10057858 0.60 TSHR (0.35) TSHRNPSR1CYP19A1
SCHEMBL709055 0.60 TSHR (0.35) TSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9802165-B2 3D expanding geometry THE UNIVERSITY OF LEEDS (GB) 2017-10-31 US disclosed
US-20140321231-A1 3D EXPANDING GEOMETRY THE UNIVERSITY OF LEEDS (GB) 2014-10-30 US disclosed