SCHEMBL16197827

SCHEMBL16197827

CC(Cl)CN1CCn2c(cc3ccccc32)C1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 16/20 0.55
HTR2A P28223 3/20 0.55
HTR2C P28335 3/20 0.55
HTR1A P08908 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13797448 0.81 HTR2A (0.75) SIGMAR1HTR2AHTR2CHTR1A
SCHEMBL16208329 0.81 SIGMAR1 (0.64) SIGMAR1HTR2AHTR2CHTR1A
SCHEMBL30585519 0.78 SIGMAR1 (0.50) SIGMAR1HTR2AHTR2CHTR1A
SCHEMBL22528277 0.78 SIGMAR1 (0.50) SIGMAR1HTR2AHTR2CHTR1A
Hydrochloric Acid SCHEMBL8986182 0.77 HTR2A (0.54) SIGMAR1HTR2AHTR2CHTR1A
SCHEMBL16208335 0.77 HTR2A (0.66) SIGMAR1HTR2AHTR2CHTR1A
Hydrochloric Acid SCHEMBL16197598 0.76 HTR2A (0.64) SIGMAR1HTR2AHTR2CHTR1A
SCHEMBL16197727 0.75 SIGMAR1 (0.58) SIGMAR1HTR2AHTR2CHTR1A
SCHEMBL16197830 0.75 SIGMAR1 (0.69) SIGMAR1HTR2AHTR2CHTR1A
SCHEMBL16197666 0.75 SIGMAR1 (0.63) SIGMAR1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2989105-A1 PYRAZINO[1,2-a]INDOLE COMPOUNDS, THEIR PREPARATION AND USE IN MEDICAMENTS Laboratorios Del. Dr. Esteve, S.A. (ES) 2016-03-02 EP disclosed
WO-2014173903-A1 PYRAZINO[1,2-a]INDOLE COMPOUNDS, THEIR PREPARATION AND USE IN MEDICAMENTS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2014-10-30 WO disclosed