SCHEMBL16199027

SCHEMBL16199027

C[C@@H]1CCN(C(=O)N[C@@H]2CCCC(Nc3nc(-c4nn(C)c5ncccc45)ncc3F)C2)C1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 1/20 0.38
HTR3A P46098 2/20 0.36
PDE5A O76074 1/20 0.35
CCNT1 O60563 1/20 0.35
CDK4 P11802 1/20 0.35
CCNA2 P20248 1/20 0.35
CCND1 P24385 1/20 0.35
CDK2 P24941 1/20 0.35
CDK9 P50750 1/20 0.35
MGLL Q99685 2/20 0.35
JAK2 O60674 1/20 0.35
JAK3 P52333 1/20 0.35
GBA1 P04062 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16199104 1.00 TLR7 (0.38) TLR7HTR3APDE5ACCNT1CDK4
SCHEMBL16199111 1.00 TLR7 (0.38) TLR7HTR3APDE5ACCNT1CDK4
SCHEMBL16199046 1.00 TLR7 (0.38) TLR7HTR3APDE5ACCNT1CDK4
SCHEMBL16199101 0.91 CCNT1 (0.38) HTR3APDE5ACCNT1CDK4CCNA2
SCHEMBL16199044 0.91 CCNT1 (0.38) HTR3APDE5ACCNT1CDK4CCNA2
SCHEMBL16199115 0.88 PDE5A (0.36) HTR3APDE5AMGLL
SCHEMBL16199045 0.88 PDE5A (0.36) HTR3APDE5AMGLL
SCHEMBL16199021 0.88 PDE5A (0.36) HTR3APDE5AMGLL
SCHEMBL16199110 0.88 PDE5A (0.36) HTR3APDE5AMGLL
SCHEMBL16199114 0.88 CCNT1 (0.35) CCNT1CDK4CCNA2CCND1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8871774-B2 Inhibitors of influenza viruses replication VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-28 US disclosed