SCHEMBL16199045

SCHEMBL16199045

C[C@@H]1CCCN1C(=O)N[C@@H]1CCCC(Nc2nc(-c3nn(C)c4ncccc34)ncc2F)C1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.36
MGLL Q99685 3/20 0.36
HTR3A P46098 1/20 0.36
GRM5 P41594 1/20 0.36
GRM1 Q13255 1/20 0.36
AURKA O14965 1/20 0.34
AURKB Q96GD4 1/20 0.34
PDE4B Q07343 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16199021 1.00 PDE5A (0.36) PDE5AMGLLHTR3AGRM5GRM1
SCHEMBL16199110 1.00 PDE5A (0.36) PDE5AMGLLHTR3AGRM5GRM1
SCHEMBL16199115 1.00 PDE5A (0.36) PDE5AMGLLHTR3AGRM5GRM1
SCHEMBL16199044 0.89 CCNT1 (0.38) PDE5AMGLLHTR3AAURKAAURKB
SCHEMBL16199101 0.89 CCNT1 (0.38) PDE5AMGLLHTR3AAURKAAURKB
SCHEMBL16199027 0.88 TLR7 (0.38) PDE5AMGLLHTR3A
SCHEMBL16199111 0.88 TLR7 (0.38) PDE5AMGLLHTR3A
SCHEMBL16199104 0.88 TLR7 (0.38) PDE5AMGLLHTR3A
SCHEMBL16199046 0.88 TLR7 (0.38) PDE5AMGLLHTR3A
SCHEMBL15400290 0.86 CDC7 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8871774-B2 Inhibitors of influenza viruses replication VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-28 US disclosed