SCHEMBL16199031

SCHEMBL16199031

Cn1cnc(C(=O)N[C@@H]2CCCC(Nc3nc(-c4n[nH]c5ncc(F)cc45)ncc3F)C2)c1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 3/20 0.39
GSK3A P49840 3/20 0.38
GSK3B P49841 3/20 0.38
JAK2 O60674 1/20 0.38
SRC P12931 1/20 0.38
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
PIK3CG P48736 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16199098 1.00 FLT3 (0.39) FLT3GSK3AGSK3BJAK2SRC
SCHEMBL15401452 0.90 SMYD3 (0.34)
SCHEMBL15399985 0.89 GRM5 (0.38) AURKAAURKB
SCHEMBL16199395 0.86 GSK3A (0.38) FLT3GSK3AGSK3BJAK2SRC
SCHEMBL16199392 0.82 GSK3A (0.41) FLT3GSK3AGSK3BJAK2SRC
SCHEMBL16199019 0.82 GSK3A (0.38) FLT3GSK3AGSK3BJAK2SRC
SCHEMBL15400687 0.82 GSK3A (0.42) FLT3GSK3AGSK3BJAK2SRC
SCHEMBL17518514 0.82 FLT3 (0.45) FLT3GSK3AGSK3BJAK2SRC
SCHEMBL15399800 0.81 GSK3A (0.39) FLT3GSK3AGSK3BJAK2SRC
SCHEMBL16199025 0.81 GSK3A (0.39) FLT3GSK3AGSK3BJAK2SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8871774-B2 Inhibitors of influenza viruses replication VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-28 US disclosed