SCHEMBL16199049

SCHEMBL16199049

Cn1nc(-c2ncc(F)c(NC3CCC[C@@H](NC(=O)C4=CCC=C4)C3)n2)c2cc(F)cnc21

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.35
AURKB Q96GD4 1/20 0.35
GSK3A P49840 3/20 0.34
GSK3B P49841 3/20 0.34
FLT3 P36888 3/20 0.34
JAK2 O60674 2/20 0.34
SRC P12931 2/20 0.34
HTR3A P46098 2/20 0.33
ROCK2 O75116 1/20 0.33
CDK2 P24941 1/20 0.33
KDR P35968 1/20 0.33
PIK3CG P48736 1/20 0.33
PLK1 P53350 1/20 0.33
ROCK1 Q13464 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16199025 0.85 GSK3A (0.39) GSK3AGSK3BFLT3JAK2SRC
SCHEMBL16199028 0.84 AURKA (0.37) AURKAAURKBGSK3AGSK3BFLT3
SCHEMBL16199071 0.76 CCNT1 (0.38) CDK2
SCHEMBL16199112 0.76 CCNT1 (0.38) CDK2
SCHEMBL16199048 0.76 CCNT1 (0.38) CDK2
SCHEMBL16199047 0.74
SCHEMBL16199102 0.74
SCHEMBL16199114 0.73 CCNT1 (0.35) CDK2
SCHEMBL16199050 0.73 CCNT1 (0.35) CDK2
SCHEMBL16199042 0.73 GSK3A (0.51) GSK3AGSK3BFLT3JAK2SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8871774-B2 Inhibitors of influenza viruses replication VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-28 US disclosed