SCHEMBL16200095

SCHEMBL16200095

CCOc1cc(C)c(F)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
MAPT P10636 4/20 0.44
TSHR P16473 1/20 0.44
PPOX P50336 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.41
RAB9A P51151 1/20 0.41
ATM Q13315 1/20 0.41
ALDH1A1 P00352 2/20 0.39
RORC P51449 1/20 0.38
HTR2C P28335 1/20 0.37
LMNA P02545 4/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HTT P42858 2/20 0.36
GAA P10253 1/20 0.36
XBP1 P17861 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19088271 0.86 PPOX (0.46) KDM4ECYP1A2CYP2C19MAPTPPOX
SCHEMBL19088273 0.84 PPOX (0.45) KDM4ECYP1A2CYP2C19MAPTPPOX
SCHEMBL30805782 0.84 KDM4E (0.51) KDM4ECYP1A2CYP2C19MAPTTSHR
SCHEMBL12129123 0.84 KDM4E (0.51) KDM4ECYP1A2CYP2C19MAPTTSHR
SCHEMBL19123074 0.82 HTT (0.45) KDM4ECYP1A2CYP2C19MAPTTSHR
SCHEMBL18304662 0.82 KDM1A (0.41) KDM4ECYP1A2CYP2C19MAPTTSHR
SCHEMBL19088275 0.80 PPOX (0.42) KDM4ECYP1A2CYP2C19MAPTPPOX
SCHEMBL8599602 0.79 PPOX (0.45) KDM4ECYP1A2CYP2C19MAPTPPOX
SCHEMBL8157623 0.79 KDM4E (0.49) KDM4ECYP1A2CYP2C19MAPTTSHR
SCHEMBL19156087 0.78 KDM1A (0.41) KDM4ECYP1A2CYP2C19MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed