SCHEMBL16200316

SCHEMBL16200316

CCc1cc(OC)c(Cl)cc1CNC1CC1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.52
MEN1 O00255 6/20 0.52
KDM4E B2RXH2 4/20 0.52
HTT P42858 3/20 0.52
GAA P10253 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
ALDH1A1 P00352 3/20 0.45
MAPT P10636 1/20 0.44
TAAR1 Q96RJ0 1/20 0.43
POLB P06746 2/20 0.41
SUV39H2 Q9H5I1 1/20 0.41
MITF O75030 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13184317 0.80 MEN1 (0.47) KMT2AMEN1KDM4EHTTGAA
SCHEMBL13184249 0.80 SLC6A4 (0.49) KDM4EGAAALDH1A1TAAR1
SCHEMBL16200315 0.78 KMT2A (0.58) KMT2AMEN1KDM4EHTTGAA
SCHEMBL13178799 0.75 KMT2A (0.55) KMT2AMEN1KDM4EHTTGAA
SCHEMBL13262991 0.73 KDM1A (0.60) KMT2AMEN1KDM4EHTTGAA
SCHEMBL19650826 0.73 KMT2A (0.57) KMT2AMEN1KDM4EHTTGAA
SCHEMBL4630869 0.72 MEN1 (0.62) KMT2AMEN1KDM4EHTTGAA
SCHEMBL737379 0.72 KMT2A (0.50) KMT2AMEN1KDM4EHTTGAA
SCHEMBL12467391 0.71 TAAR1 (0.53) KDM4EGAAALDH1A1MAPTTAAR1
SCHEMBL21233362 0.71 TAAR1 (0.53) KDM4EGAAALDH1A1MAPTTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed