SCHEMBL16201142

SCHEMBL16201142

Cc1nnc(C(C)C)n1C1CC2CCC(C1)N2CC[C@H](NC(=O)C1CCC(C)(C)CC1)c1ccccc1

nearest known ligand 0.88

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 20/20 0.88
KCNH2 Q12809 7/20 0.88
CYP3A4 P08684 2/20 0.88
ADRA2A P08913 1/20 0.88
CYP2C9 P11712 1/20 0.88
KCNE1 P15382 1/20 0.88
OPRM1 P35372 1/20 0.88
KCNQ1 P51787 1/20 0.88
SLC47A1 Q96FL8 1/20 0.88

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maraviroc SCHEMBL4576508 0.93 CCR5 (1.00) CCR5KCNH2CYP3A4ADRA2ACYP2C9
Maraviroc SCHEMBL51991 0.93 CCR5 (1.00) CCR5KCNH2CYP3A4ADRA2ACYP2C9
Maraviroc SCHEMBL334506 0.93 CCR5 (1.00) CCR5KCNH2CYP3A4ADRA2ACYP2C9
Maraviroc SCHEMBL12611449 0.93 CCR5 (1.00) CCR5KCNH2CYP3A4ADRA2ACYP2C9
Maraviroc SCHEMBL20451355 0.93 CCR5 (1.00) CCR5KCNH2CYP3A4ADRA2ACYP2C9
Maraviroc SCHEMBL1053748 0.93 CCR5 (1.00) CCR5KCNH2CYP3A4ADRA2ACYP2C9
Maraviroc SCHEMBL2177194 0.93 CCR5 (1.00) CCR5KCNH2CYP3A4ADRA2ACYP2C9
SCHEMBL15375827 0.92 CCR5 (0.84) CCR5KCNH2CYP3A4ADRA2ACYP2C9
SCHEMBL3876067 0.92 CCR5 (0.84) CCR5KCNH2CYP3A4ADRA2ACYP2C9
SCHEMBL15375694 0.92 CCR5 (0.84) CCR5KCNH2CYP3A4ADRA2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014173375-A1 A PROCESS FOR THE SYNTHESIS OF MARAVIROC ZENTIVA, K.S. (CZ) 2014-10-30 WO disclosed