SCHEMBL16202189

SCHEMBL16202189

C#CCC[C@@H](NC(=O)OC(C)(C)C)[C@@H](O)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSK P43235 7/20 0.49
CTSS P25774 6/20 0.49
KLK5 Q9Y337 2/20 0.43
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
MAPT P10636 1/20 0.42
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16202188 1.00 CTSK (0.49) CTSKCTSSKLK5CTSLCTSB
SCHEMBL16202186 1.00 CTSK (0.49) CTSKCTSSKLK5CTSLCTSB
SCHEMBL16119982 1.00 CTSK (0.49) CTSKCTSSKLK5CTSLCTSB
SCHEMBL14971377 1.00 CTSK (0.49) CTSKCTSSKLK5CTSLCTSB
SCHEMBL20085530 0.88 CTSK (0.51) CTSKCTSSKLK5CTSLCTSB
SCHEMBL14971379 0.87 AOC3 (0.42) MAPT
SCHEMBL21336988 0.87 AOC3 (0.42) MAPT
SCHEMBL21336975 0.87 AOC3 (0.42) MAPT
SCHEMBL21336985 0.87 AOC3 (0.42) MAPT
SCHEMBL21336987 0.87 AOC3 (0.42) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240018489-A1 BIOCATALYSTS FOR THE PREPARATION OF HYDROXY SUBSTITUTED CARBAMATES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2024-01-18 US disclosed
US-20240018489-A1 BIOCATALYSTS FOR THE PREPARATION OF HYDROXY SUBSTITUTED CARBAMATES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2024-01-18 US disclosed
US-11713451-B2 Biocatalysts for the preparation of hydroxy substituted carbamates CODEXIS, INC. (US) 2023-08-01 US disclosed
US-11713451-B2 Biocatalysts for the preparation of hydroxy substituted carbamates CODEXIS, INC. (US) 2023-08-01 US disclosed
US-20210071151-A1 BIOCATALYSTS FOR THE PREPARATION OF HYDROXY SUBSTITUTED CARBAMATES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2021-03-11 US disclosed
US-10851351-B2 Biocatalysts for the preparation of hydroxy substituted carbamates CODEXIS, INC. (US) 2020-12-01 US disclosed
US-10253303-B2 Biocatalysts for the preparation of hydroxy substituted carbamates CODEXIS, INC. (US) 2019-04-09 US disclosed
US-20180010100-A1 BIOCATALYSTS FOR THE PREPARATION OF HYDROXY SUBSTITUTED CARBAMATES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2018-01-11 US disclosed
US-9803178-B2 Biocatalysts for the preparation of hydroxy substituted carbamates CODEXIS, INC. (US) 2017-10-31 US disclosed
US-9803178-B2 Biocatalysts for the preparation of hydroxy substituted carbamates CODEXIS, INC. (US) 2017-10-31 US disclosed
US-20160319247-A1 BIOCATALYSTS FOR THE PREPARATION OF HYDROXY SUBSTITUTED CARBAMATES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2016-11-03 US disclosed
US-20160319247-A1 BIOCATALYSTS FOR THE PREPARATION OF HYDROXY SUBSTITUTED CARBAMATES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2016-11-03 US disclosed
US-9422531-B2 Biocatalysts for the preparation of hydroxy substituted carbamates CODEXIS, INC. (US) 2016-08-23 US disclosed
US-9422531-B2 Biocatalysts for the preparation of hydroxy substituted carbamates CODEXIS, INC. (US) 2016-08-23 US disclosed
US-20150344850-A1 BIOCATALYSTS FOR THE PREPARATION OF HYDROXY SUBSTITUTED CARBAMATES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2015-12-03 US disclosed
US-20150344850-A1 BIOCATALYSTS FOR THE PREPARATION OF HYDROXY SUBSTITUTED CARBAMATES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2015-12-03 US disclosed
US-9139819-B2 Biocatalysts for the preparation of hydroxy substituted carbamates CODEXIS, INC. (US) 2015-09-22 US disclosed
US-9139819-B2 Biocatalysts for the preparation of hydroxy substituted carbamates CODEXIS, INC. (US) 2015-09-22 US disclosed
US-20140322769-A1 BIOCATALYSTS FOR THE PREPARATION OF HYDROXY SUBSTITUTED CARBAMATES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2014-10-30 US disclosed
US-20140322769-A1 BIOCATALYSTS FOR THE PREPARATION OF HYDROXY SUBSTITUTED CARBAMATES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2014-10-30 US disclosed