SCHEMBL16208754

SCHEMBL16208754

N[C@H](C(=O)Cl)[C@H](O)c1ccc2c(c1)OCO2

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 2/20 0.45
MAPK9 P45984 1/20 0.44
ALDH1A1 P00352 2/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
HPGD P15428 1/20 0.42
AOC3 Q16853 1/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
LMNA P02545 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
SLC6A4 P31645 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5279500 0.86 PTGS1 (0.55) EDNRAMAPK9ALDH1A1MAPK1KMT2A
SCHEMBL7433780 0.86 PTGS1 (0.55) EDNRAMAPK9ALDH1A1MAPK1KMT2A
SCHEMBL16208746 0.86 PTGS1 (0.55) EDNRAMAPK9ALDH1A1MAPK1KMT2A
Acetic Acid SCHEMBL10875129 0.82 PTGS1 (0.51) EDNRAMAPK9ALDH1A1MAPK1KMT2A
Acetic Acid SCHEMBL10942103 0.82 PTGS1 (0.51) EDNRAMAPK9ALDH1A1MAPK1KMT2A
SCHEMBL10874124 0.81 EDNRA (0.51) EDNRAALDH1A1KMT2AMEN1HPGD
SCHEMBL18076242 0.81 EDNRA (0.51) EDNRAALDH1A1KMT2AMEN1HPGD
SCHEMBL10875005 0.81 EDNRA (0.51) EDNRAALDH1A1KMT2AMEN1HPGD
Hydrochloric Acid SCHEMBL10874331 0.80 EDNRA (0.50) EDNRAKMT2AMEN1HPGD
SCHEMBL7898797 0.80 CYP3A4 (0.54) MAPK9ALDH1A1MAPK1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014174425-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ORTHOSTASIS AND NEUROLOGICAL DISEASES KANDULA MAHESH (IN) 2014-10-30 WO disclosed