SCHEMBL7898797

SCHEMBL7898797

OC(c1ccc2c(c1)OCO2)C(O)c1ccc2c(c1)OCO2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.54
CYP2D6 P10635 3/20 0.51
MAPK1 P28482 2/20 0.51
CYP1A2 P05177 2/20 0.51
CYP2C9 P11712 2/20 0.51
CYP2C19 P33261 2/20 0.51
SMAD3 P84022 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
AOC3 Q16853 1/20 0.49
P4HB P07237 2/20 0.47
MAPK9 P45984 1/20 0.47
ACHE P22303 2/20 0.47
PGR P06401 1/20 0.47
AR P10275 1/20 0.47
GABRA1 P14867 1/20 0.47
MAOA P21397 1/20 0.47
SLC6A2 P23975 1/20 0.47
PDE4A P27815 1/20 0.47
KDR P35968 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2608968 0.90 MEN1 (0.52) CYP3A4CYP2D6MAPK1CYP1A2CYP2C9
SCHEMBL10931500 0.88 MEN1 (0.51) CYP3A4CYP2D6MAPK1CYP1A2CYP2C9
SCHEMBL1599758 0.87 CYP3A4 (0.54) CYP3A4CYP2D6MAPK1CYP1A2CYP2C9
SCHEMBL18626121 0.87 CYP3A4 (0.54) CYP3A4CYP2D6MAPK1CYP1A2CYP2C9
SCHEMBL11423964 0.85 TAAR1 (0.54) CYP3A4CYP2D6CYP1A2CYP2C9CYP2C19
SCHEMBL9799615 0.85 CYP3A4 (0.53) CYP3A4CYP2D6MAPK1CYP1A2CYP2C9
SCHEMBL7990464 0.84 MAPK9 (0.54) CYP3A4CYP2D6MAPK1CYP1A2CYP2C9
SCHEMBL29664492 0.83 KMT2A (0.54) CYP3A4CYP2D6MAPK1CYP1A2CYP2C9
SCHEMBL1155200 0.83 KMT2A (0.54) CYP3A4CYP2D6MAPK1CYP1A2CYP2C9
SCHEMBL13882955 0.82 CYP3A4 (0.50) CYP3A4CYP2D6MAPK1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6194019-B1 ORGANOLEPTIC 1,2-DIOL DISUBSTITUTED WITH PHENYL, CYCLOHEXYL, OR BENZODIOXOLE RINGS; FOODS, TOBACCO; MASKING SMOKE ODORS GIVAUDAN S.A. (CH) 2001-02-27 US claimed
EP-0746986-B1 Delayed release flavourant compositions GIVAUDAN ROURE INT (CH) 2000-08-23 EP claimed
US-5904148-A Delayed release flavorant compositions GIVADUAN-ROURE (INTERNATIONAL) SA (CH) 1999-05-18 US claimed
EP-0746986-A2 Delayed release flavourant compositions GIVAUDAN-ROURE (INTERNATIONAL) S.A. (CH) 1996-12-11 EP claimed
US-6194019-B1 ORGANOLEPTIC 1,2-DIOL DISUBSTITUTED WITH PHENYL, CYCLOHEXYL, OR BENZODIOXOLE RINGS; FOODS, TOBACCO; MASKING SMOKE ODORS GIVAUDAN S.A. (CH) 2001-02-27 US disclosed
EP-0746986-B1 Delayed release flavourant compositions GIVAUDAN ROURE INT (CH) 2000-08-23 EP disclosed
US-5921247-A Delayed release flavorant compositions GIVAUDAN-ROURE (INTERNATIONAL) SA (CH) 1999-07-13 US disclosed
US-5904148-A Delayed release flavorant compositions GIVADUAN-ROURE (INTERNATIONAL) SA (CH) 1999-05-18 US disclosed
EP-0746986-A2 Delayed release flavourant compositions GIVAUDAN-ROURE (INTERNATIONAL) S.A. (CH) 1996-12-11 EP disclosed