SCHEMBL16214701

SCHEMBL16214701

CCOc1ccc(C#Cc2ccc(C(C)C(=O)Nc3ccccc3)cc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ACACB O00763 18/20 0.57
GPR88 Q9GZN0 1/20 0.55
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16214704 0.84 ACACB (0.57) ACACB
SCHEMBL16214700 0.83 ACACB (0.64) ACACB
SCHEMBL458764 0.81 AKR1C3 (0.64) ACACB
SCHEMBL16214698 0.78 ACACB (0.60) ACACBGPR88
SCHEMBL16214695 0.77 SMN1; SMN2 (0.60) ACACBNPC1RAB9A
SCHEMBL462647 0.76 ACACB (0.50) ACACB
SCHEMBL7748974 0.76 POLB (0.66)
SCHEMBL17365594 0.76 POLB (0.66)
SCHEMBL7472046 0.75 NPC1 (0.58) NPC1RAB9A
SCHEMBL18119719 0.73 MAPT (0.67) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614054-B1 ETHYNE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INT (DE) 2014-11-19 EP disclosed
US-8877754-B2 Compounds, pharmaceutical compositions and uses thereof BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-11-04 US disclosed