SCHEMBL16215902

SCHEMBL16215902

CN(C)Cc1cc2ccccc2cn1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CYP2A6 P11509 1/20 0.48
ATM Q13315 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
PDPK1 O15530 1/20 0.44
PDE10A Q9Y233 4/20 0.41
TRPM8 Q7Z2W7 1/20 0.40
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 1/20 0.39
CXCR4 P61073 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
HTR3A P46098 1/20 0.38
CYP2D6 P10635 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
PLAU P00749 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12088909 0.82 ATM (0.46) CYP1A2CYP2A6ATML3MBTL1PDPK1
SCHEMBL13792017 0.81 MAPT (0.50) CYP1A2CYP2A6ATML3MBTL1PDPK1
SCHEMBL4367341 0.78 ATM (0.45) CYP1A2CYP2A6ATML3MBTL1PDPK1
SCHEMBL873512 0.78 CYP1A2 (0.54) CYP1A2CYP2A6ATML3MBTL1PDPK1
SCHEMBL14274065 0.75 CYP1A2 (0.47) CYP1A2CYP2A6ATML3MBTL1PDPK1
SCHEMBL6114924 0.74 ATM (0.57) CYP1A2CYP2A6ATML3MBTL1PDPK1
SCHEMBL3823640 0.74 ATM (0.51) CYP1A2CYP2A6ATML3MBTL1PDPK1
SCHEMBL13977557 0.74 ATM (0.51) CYP1A2CYP2A6ATML3MBTL1PDPK1
SCHEMBL3639574 0.74 PDPK1 (0.54) CYP1A2CYP2A6ATML3MBTL1PDPK1
SCHEMBL2908675 0.74 L3MBTL1 (0.51) CYP1A2CYP2A6ATML3MBTL1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2470012-B1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME (US) 2014-11-05 EP disclosed