SCHEMBL16217181

SCHEMBL16217181

Clc1ccc2c(n1)CN(Cc1ccccc1)CC2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.56
KMT2A Q03164 3/20 0.56
MEN1 O00255 2/20 0.56
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
DHFR P00374 1/20 0.49
C5AR1 P21730 1/20 0.48
SIGMAR1 Q99720 4/20 0.46
DRD4 P21917 2/20 0.46
HTR2B P41595 2/20 0.46
TMEM97 Q5BJF2 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
ADRA2A P08913 1/20 0.46
ADRA2B P18089 1/20 0.46
HRH1 P35367 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30474228 1.00 PNMT (0.56) PNMTKMT2AMEN1NPC1RAB9A
SCHEMBL29883119 0.88 KMT2A (0.63) PNMTKMT2AMEN1NPC1RAB9A
SCHEMBL1038680 0.88 KMT2A (0.63) PNMTKMT2AMEN1NPC1RAB9A
SCHEMBL16217183 0.84 MEN1 (0.54) PNMTKMT2AMEN1NPC1RAB9A
SCHEMBL30474206 0.84 KMT2A (0.54) PNMTKMT2AMEN1NPC1RAB9A
SCHEMBL30474287 0.84 KMT2A (0.54) PNMTKMT2AMEN1NPC1RAB9A
SCHEMBL16220548 0.84 KMT2A (0.54) PNMTKMT2AMEN1NPC1RAB9A
SCHEMBL16217185 0.82 PNMT (0.52) PNMTKMT2AMEN1NPC1RAB9A
SCHEMBL16210349 0.81 KMT2A (0.51) PNMTKMT2AMEN1NPC1RAB9A
SCHEMBL19042312 0.81 MEN1 (0.51) PNMTKMT2AMEN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250109148-A1 HETEROCYCLIC GLP-1 AGONISTS SHANGHAI SHOUTI BIOTECHNOLOGY CO., LTD. (CN) 2025-04-03 US disclosed
EP-2991989-B1 IMIDAZO-TRIAZINE DERIVATIVES AS PDE10 INHIBITORS PFIZER (US) 2017-06-28 EP disclosed
US-9296761-B2 Triazine derivatives PFIZER INC. (US) 2016-03-29 US disclosed
US-9296761-B2 Triazine derivatives PFIZER INC. (US) 2016-03-29 US disclosed
US-20150353579-A1 Triazine Derivatives PFIZER (US) 2015-12-10 US disclosed
US-20150353579-A1 Triazine Derivatives PFIZER (US) 2015-12-10 US disclosed
US-9145427-B2 Triazine derivatives PFIZER INC. (US) 2015-09-29 US disclosed
US-9145427-B2 Triazine derivatives PFIZER INC. (US) 2015-09-29 US disclosed
US-20150080401-A1 Triazine Derivatives PFIZER (US) 2015-03-19 US disclosed
US-20150080401-A1 Triazine Derivatives PFIZER (US) 2015-03-19 US disclosed
US-8933224-B2 Triazine derivatives PFIZER INC. (US) 2015-01-13 US disclosed
US-8933224-B2 Triazine derivatives PFIZER INC. (US) 2015-01-13 US disclosed
US-20140329820-A1 Triazine Derivatives PFIZER INC. (US) 2014-11-06 US disclosed
US-20140329820-A1 Triazine Derivatives PFIZER INC. (US) 2014-11-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140329820-A1 Triazine Derivatives PDE12, PDE5A, PDE10A PNMT 750/4885KMT2A 1941/4885MEN1 3132/4885
US-20250109148-A1 HETEROCYCLIC GLP-1 AGONISTS GLP1R, GIPR, GCGR PNMT 2301/4885KMT2A 3670/4885MEN1 450/4885
US-20150353579-A1 Triazine Derivatives PDE12, PDE5A, PDE10A PNMT 750/4885KMT2A 1941/4885MEN1 3132/4885
US-20150080401-A1 Triazine Derivatives PDE12, PDE5A, PDE10A PNMT 750/4885KMT2A 1941/4885MEN1 3132/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.