SCHEMBL16224064

SCHEMBL16224064

CC(C)(C)NC(=O)O[C@H]1CC[C@H](N)CC1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.37
DPP4 P27487 2/20 0.35
CCNE1 P24864 12/20 0.34
CDK2 P24941 12/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
GSK3B P49841 7/20 0.33
SMYD3 Q9H7B4 1/20 0.33
APOBEC3A P31941 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2145078 1.00 EPHX1 (0.37) EPHX1DPP4CCNE1CDK2SMN1; SMN2
SCHEMBL2145085 1.00 EPHX1 (0.37) EPHX1DPP4CCNE1CDK2SMN1; SMN2
SCHEMBL25270786 0.93 EPHX1 (0.40) EPHX1DPP4CCNE1CDK2SMN1; SMN2
SCHEMBL27855976 0.91 NAAA (0.35) EPHX1DPP4CCNE1CDK2GSK3B
SCHEMBL7815595 0.90 EPHX1 (0.42) EPHX1DPP4CCNE1CDK2SMN1; SMN2
SCHEMBL23437012 0.89 EPHX1 (0.42) EPHX1DPP4SMN1; SMN2APOBEC3AAPOBEC3G
SCHEMBL25281021 0.89 CCNE1 (0.37) DPP4CCNE1CDK2GSK3B
SCHEMBL25271862 0.89 CCNE1 (0.37) DPP4CCNE1CDK2GSK3B
SCHEMBL27760444 0.89 CCNE1 (0.37) DPP4CCNE1CDK2GSK3B
Methane SCHEMBL27968861 0.88 EPHX1 (0.41) EPHX1DPP4CCNE1CDK2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108727363-B Novel cyclin dependent kinase CDK9 inhibitor 劲方医药科技(上海)有限公司 2020-06-19 CN disclosed
EP-2470536-B1 Methylpyrrolopyrimidinecarboxamides TAKEDA GMBH (DE) 2014-11-12 EP disclosed