SCHEMBL16237462

SCHEMBL16237462

CC(C)(C)OC(=O)c1c(Nc2c(C(=O)O)sc3cnccc23)ccc(F)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
CASP1 P29466 1/20 0.39
HTT P42858 1/20 0.39
CASP7 P55210 1/20 0.39
NCOA1 Q15788 1/20 0.39
HSD17B10 Q99714 1/20 0.39
RCE1 Q9Y256 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
RPS6KB1 P23443 1/20 0.35
CDK2 P24941 1/20 0.35
MAPKAPK2 P49137 1/20 0.35
GSK3B P49841 1/20 0.35
RPS6KA3 P51812 1/20 0.35
ACVR1B P36896 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723555 0.77 ALDH1A1 (0.50) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL3997430 0.72 MAP2K1 (0.48) IDO1
SCHEMBL4003188 0.72 GAA (0.44) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL16237538 0.68 CSNK2A1 (0.54) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL14230457 0.67 ALDH1A1 (0.46) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL16237464 0.67 HTT (0.35) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL3642155 0.67 MCL1 (0.60) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL1218574 0.66 MAP2K1 (0.47) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL1216500 0.66 MAP2K1 (0.44) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL4723937 0.65 ALDH1A1 (0.42) ALDH1A1KDM4EGLAGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970173-B1 INHIBITORS OF THE KYNURENINE PATHWAY CURADEV PHARMA PRIVATE LTD (IN) 2018-05-09 EP disclosed
EP-2970173-A1 INHIBITORS OF THE KYNURENINE PATHWAY Curadev Pharma Private Ltd. (IN) 2016-01-20 EP disclosed
WO-2014186035-A1 INHIBITORS OF THE KYNURENINE PATHWAY CURADEV PHARMA PRIVATE LTD. (IN) 2014-11-20 WO disclosed