SCHEMBL16237698

SCHEMBL16237698

O=C(O)c1c(CBr)nc(-c2nccs2)nc1-c1ccc(F)c(F)c1Cl

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.33
ECE1 P42892 1/20 0.32
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
EIF4E P06730 2/20 0.30
KMO O15229 1/20 0.30
CTSA P10619 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16237062 0.90 ECE1 (0.34) ADORA2AECE1EIF4ECTSA
SCHEMBL16237173 0.88 CTSA (0.41) ADORA2AECE1HDAC3HDAC1HDAC6
SCHEMBL16237487 0.84 HDAC3 (0.43) ADORA2AHDAC3HDAC1HDAC6EIF4E
SCHEMBL16237675 0.83 ADORA2A (0.39) ADORA2AECE1CTSA
SCHEMBL17064231 0.82 KMT2A (0.40) ADORA2AECE1HDAC3HDAC1HDAC6
SCHEMBL16237522 0.81 HDAC3 (0.36) ADORA2AECE1HDAC3HDAC1HDAC6
SCHEMBL16237804 0.81 KMO (0.38) ADORA2AECE1HDAC3HDAC1HDAC6
SCHEMBL16237622 0.80 KMO (0.41) ADORA2AEIF4EKMO
SCHEMBL17064250 0.80 HCRTR1 (0.39) ADORA2AECE1CTSA
SCHEMBL16236743 0.79 ADORA2A (0.39) ADORA2AECE1HDAC3HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2997032-A1 6-BRIDGED HETEROARYLDIHYDROPYRIMIDINES FOR THE TREATMENT AND PROPHYLAXIS OF HEPATITIS B VIRUS INFECTION F. Hoffmann-La Roche AG (CH) 2016-03-23 EP disclosed
WO-2014184328-A1 6-BRIDGED HETEROARYLDIHYDROPYRIMIDINES FOR THE TREATMENT AND PROPHYLAXIS OF HEPATITIS B VIRUS INFECTION F. HOFFMANN-LA ROCHE AG (CH) 2014-11-20 WO disclosed