SCHEMBL16239587

SCHEMBL16239587

C[C@@]1(CNC(=O)O)CN(C(=O)c2ccc(C#N)cc2)C[C@H]1c1ccc(Cl)cc1

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 16/20 0.65
ALDH1A1 P00352 1/20 0.42
ITGB2 P05107 2/20 0.41
ICAM1 P05362 2/20 0.41
ITGAL P20701 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16239760 0.87 TACR3 (0.72) TACR3
SCHEMBL16239531 0.85 TACR3 (0.57) TACR3
SCHEMBL16239680 0.82 TACR3 (0.70) TACR3
SCHEMBL16239928 0.80 TACR3 (0.70) TACR3
SCHEMBL16240045 0.79 TACR3 (0.69) TACR3ALDH1A1
SCHEMBL16239851 0.79 TACR3 (0.70) TACR3
SCHEMBL322188 0.79 TACR3 (1.00) TACR3
SCHEMBL10026138 0.79 TACR3 (1.00) TACR3
SCHEMBL16239590 0.78 TACR3 (0.72) TACR3ALDH1A1ITGB2ICAM1ITGAL
SCHEMBL16239696 0.77 TACR3 (0.53) TACR3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2661432-B1 PYRROLIDINE DERIVATIVES AS NK3 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2014-11-19 EP claimed