SCHEMBL16239696

SCHEMBL16239696

C[C@@]1(c2ccc(Cl)cc2)CN(C(=O)c2ccc(C#N)cc2)C[C@@H]1CNC(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 5/20 0.53
ALDH1A1 P00352 1/20 0.42
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
PGGT1B P53609 1/20 0.39
PTGER4 P35408 1/20 0.39
PTGER2 P43116 1/20 0.39
PTGDR Q13258 1/20 0.39
NR1H4 Q96RI1 2/20 0.38
HCRTR2 O43614 1/20 0.38
NR1I2 O75469 1/20 0.37
RORC P51449 1/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
FASN P49327 4/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
GFER P55789 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16239535 0.80 TACR3 (0.57) TACR3ALDH1A1MAPT
SCHEMBL16239697 0.78 TACR3 (0.72) TACR3ALDH1A1NR1H4HCRTR2
SCHEMBL16239587 0.77 TACR3 (0.65) TACR3ALDH1A1
SCHEMBL16239847 0.74 TACR3 (0.53) TACR3NR1I2RORC
SCHEMBL16239718 0.72 CCR3 (0.43) NR1I2RORC
SCHEMBL16239921 0.72 TACR3 (0.55) TACR3NR1I2RORC
SCHEMBL16239791 0.72 TACR3 (0.56) TACR3
SCHEMBL10277847 0.70 TACR3 (1.00) TACR3
SCHEMBL16239590 0.69 TACR3 (0.72) TACR3ALDH1A1
SCHEMBL16239565 0.67 TACR3 (0.60) TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2661432-B1 PYRROLIDINE DERIVATIVES AS NK3 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2014-11-19 EP claimed