SCHEMBL16248161

SCHEMBL16248161

CCOCCCc1cccc(C)c1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.52
IDO1 P14902 2/20 0.46
HRH3 Q9Y5N1 3/20 0.44
KCNH2 Q12809 2/20 0.43
DAO P14920 1/20 0.43
CYP4F2 P78329 1/20 0.42
CYP4A11 Q02928 1/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
GPR84 Q9NQS5 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
LTB4R Q15722 1/20 0.40
LTB4R2 Q9NPC1 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22480217 0.95 TAAR1 (0.50) TAAR1IDO1HRH3DAOCYP4F2
SCHEMBL10204846 0.89 TAAR1 (0.55) TAAR1IDO1HRH3KCNH2DAO
SCHEMBL14234021 0.84 CYP4F2 (0.43) IDO1KCNH2CYP4F2CYP4A11ALDH1A1
SCHEMBL15432887 0.83 TAAR1 (0.49) TAAR1IDO1HRH3KCNH2DAO
SCHEMBL12136331 0.81 TAAR1 (0.55) TAAR1IDO1HRH3DAOALDH1A1
SCHEMBL20463165 0.81 SMN1; SMN2 (0.40) TAAR1IDO1CYP4F2CYP4A11ALDH1A1
SCHEMBL8092500 0.80 TAAR1 (0.68) TAAR1IDO1HRH3DAOGPR84
SCHEMBL8099771 0.80 TAAR1 (0.68) TAAR1IDO1HRH3DAOGPR84
SCHEMBL14228549 0.80 IDO1 (0.56) TAAR1IDO1ALDH1A1CYP2D6
SCHEMBL167733 0.79 TAAR1 (0.61) TAAR1IDO1HRH3DAORAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9079918-B2 Macrocycles as factor XIa inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2015-07-14 US disclosed
US-20140343276-A1 MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2014-11-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140343276-A1 MACROCYCLES AS FACTOR XIA INHIBITORS TFPI, TFPI2, F11 TAAR1 4566/4885IDO1 2082/4885HRH3 1723/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.