SCHEMBL1624888

SCHEMBL1624888

O=C(Nc1cccc(-c2nc(-c3ccccc3)c[nH]2)c1)c1ccc(N2CCCCCC2)nc1.O=C(Nc1cccc(-c2ncc(-c3ccccc3)[nH]2)c1)c1ccc(N2CCOCC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 10/20 0.50
RAB9A P51151 10/20 0.50
ATR Q13535 2/20 0.43
TRPV1 Q8NER1 1/20 0.42
AURKA O14965 1/20 0.42
KDR P35968 1/20 0.42
FLT3 P36888 1/20 0.42
DGAT1 O75907 1/20 0.42
BTK Q06187 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1625212 0.88 NPC1 (0.60) NPC1RAB9AATRDGAT1
SCHEMBL1624353 0.87 TRPV1 (0.51) NPC1RAB9ATRPV1AURKA
SCHEMBL1625531 0.87 TRPV1 (0.51) NPC1RAB9ATRPV1AURKA
SCHEMBL1624266 0.84 NPC1 (0.60) NPC1RAB9AATRAURKAKDR
SCHEMBL1625249 0.84 NPC1 (0.55) NPC1RAB9AATRAURKAKDR
Benzamide SCHEMBL27756821 0.84 NPC1 (0.43) NPC1RAB9AATRAURKAKDR
SCHEMBL1623276 0.80 KCNQ3 (0.56) NPC1RAB9AATRDGAT1
SCHEMBL1625106 0.73 HDAC1 (0.46) NPC1RAB9AATRDGAT1BTK
SCHEMBL1623219 0.73 MTOR (0.53) NPC1RAB9A
SCHEMBL1623606 0.73 RAF1 (0.55) NPC1RAB9ADGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7928133-B2 Compounds and compositions as hedgehog signaling pathway modulators IRM LLC (BM) 2011-04-19 US claimed