SCHEMBL1625531

SCHEMBL1625531

O=C(Nc1cccc(-c2nc(-c3ccccc3)c[nH]2)c1)c1ccc(N2CCCCCC2)nc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.51
CNR1 P21554 6/20 0.50
NPC1 O15118 7/20 0.48
RAB9A P51151 7/20 0.48
KCNH2 Q12809 1/20 0.46
KCNQ3 O43525 1/20 0.46
KCNQ2 O43526 1/20 0.46
MCHR1 Q99705 1/20 0.45
AURKA O14965 1/20 0.45
RPS6KB1 P23443 1/20 0.45
AURKB Q96GD4 1/20 0.45
PAX8 Q06710 1/20 0.45
KMT2A Q03164 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC2 Q92769 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1624353 1.00 TRPV1 (0.51) TRPV1CNR1NPC1RAB9AKCNH2
SCHEMBL1625212 0.91 NPC1 (0.60) NPC1RAB9A
SCHEMBL1624888 0.87 NPC1 (0.50) TRPV1NPC1RAB9AAURKA
SCHEMBL1624770 0.82 HDAC2 (0.45) TRPV1KCNH2MCHR1HDAC3HDAC2
SCHEMBL1624235 0.82 HDAC2 (0.45) TRPV1KCNH2MCHR1HDAC3HDAC2
SCHEMBL1623276 0.81 KCNQ3 (0.56) NPC1RAB9AKCNQ3KCNQ2
SCHEMBL27696834 0.80 MCHR1 (0.60) TRPV1NPC1RAB9AKCNQ3KCNQ2
SCHEMBL6925885 0.79 CNR2 (0.56) CNR1NPC1RAB9AKMT2A
SCHEMBL1624266 0.79 NPC1 (0.60) NPC1RAB9AAURKA
SCHEMBL6925668 0.78 CNR2 (0.53) CNR1NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090312308-A1 COMPOUNDS AND COMPOSITIONS AS HEDGEHOG SIGNALING PATHWAY MODULATORS IRM LLC (BM) 2009-12-17 US claimed
US-7928133-B2 Compounds and compositions as hedgehog signaling pathway modulators IRM LLC (BM) 2011-04-19 US disclosed
US-7928133-B2 Compounds and compositions as hedgehog signaling pathway modulators IRM LLC (BM) 2011-04-19 US disclosed
US-7928133-B2 Compounds and compositions as hedgehog signaling pathway modulators IRM LLC (BM) 2011-04-19 US disclosed
US-20090312308-A1 COMPOUNDS AND COMPOSITIONS AS HEDGEHOG SIGNALING PATHWAY MODULATORS IRM LLC (BM) 2009-12-17 US disclosed
US-20090312308-A1 COMPOUNDS AND COMPOSITIONS AS HEDGEHOG SIGNALING PATHWAY MODULATORS IRM LLC (BM) 2009-12-17 US disclosed
US-20090312308-A1 COMPOUNDS AND COMPOSITIONS AS HEDGEHOG SIGNALING PATHWAY MODULATORS IRM LLC (BM) 2009-12-17 US disclosed
WO-2008014291-A2 COMPOUNDS AND COMPOSITIONS AS HEDGEHOG SIGNALING PATHWAY MODULATORS IRM LLC (BM) 2008-01-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090312308-A1 COMPOUNDS AND COMPOSITIONS AS HEDGEHOG SIGNALING PATHWAY MODULATORS GLI1, SHH, SMO TRPV1 4134/4885CNR1 2415/4885NPC1 792/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.