SCHEMBL16254262

SCHEMBL16254262

Cc1c(Cc2c(Cl)cccc2Cl)c(=O)oc2cc(OCC(=O)OCC(=O)c3ccc(Cl)cc3)ccc12

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.66
CA9 Q16790 4/20 0.66
ALDH1A1 P00352 12/20 0.60
KDM4E B2RXH2 11/20 0.60
HPGD P15428 9/20 0.60
SMN1; SMN2 Q16637 4/20 0.60
LMNA P02545 1/20 0.54
MEN1 O00255 5/20 0.54
KMT2A Q03164 5/20 0.54
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
POLB P06746 1/20 0.54
HSD17B10 Q99714 5/20 0.52
ATM Q13315 1/20 0.51
HTT P42858 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
MAPT P10636 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14027239 0.74 KDM4E (0.63) CA12CA9ALDH1A1KDM4EHPGD
SCHEMBL18095545 0.73 CA9 (0.83) CA12CA9ALDH1A1KDM4EHPGD
SCHEMBL7860297 0.73 AKR1C3 (0.68) CA12CA9ALDH1A1KDM4EHPGD
SCHEMBL20554014 0.72 CA12 (0.83) CA12CA9ALDH1A1KDM4EHPGD
SCHEMBL5646958 0.72 HSD17B3 (0.69) ALDH1A1KDM4EHPGDHSD17B10NPSR1
SCHEMBL18095375 0.72 ALDH1A1 (0.72) CA12CA9ALDH1A1KDM4EHPGD
SCHEMBL18095542 0.72 CA12 (0.71) CA12CA9ALDH1A1KDM4EHPGD
SCHEMBL29527472 0.71 ALDH1A1 (0.68) ALDH1A1KDM4EHPGDSMN1; SMN2LMNA
SCHEMBL5647066 0.71 MAP2K1 (0.58) ALDH1A1KDM4EHPGDSMN1; SMN2MEN1
SCHEMBL5648696 0.71 MAP2K1 (0.53) ALDH1A1KDM4EHPGDSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170003275-A1 METHOD TO IDENTIFY COMPOUNDS ABLE TO BIND TO THE ROSSMANN FOLD OF C-TERMINAL-BINDING PROTEINS, IDENTIFIED COMPOUNDS AND MEDICAL USES THEREOF CONSIGLIO NAZIONALE DELLE RICERCHE (IT) 2017-01-05 US disclosed
US-20170003275-A1 METHOD TO IDENTIFY COMPOUNDS ABLE TO BIND TO THE ROSSMANN FOLD OF C-TERMINAL-BINDING PROTEINS, IDENTIFIED COMPOUNDS AND MEDICAL USES THEREOF CONSIGLIO NAZIONALE DELLE RICERCHE (IT) 2017-01-05 US disclosed
WO-2014184370-A1 METHOD TO IDENTIFY COMPOUNDS ABLE TO BIND TO THE ROSSMANN FOLD OF C-TERMINAL-BINDING PROTEINS, IDENTIFIED COMPOUNDS AND MEDICAL USES THEREOF CONSIGLIO NAZIONALE DELLE RICERCHE (IT) 2014-11-20 WO disclosed