SCHEMBL16258372

SCHEMBL16258372

C=C1CC2(CCC2)Cc2nc(Cl)c(C(=O)OCC)c(O)c21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.37
GAA P10253 3/20 0.36
HTT P42858 1/20 0.36
CYP1A2 P05177 3/20 0.34
CYP2C9 P11712 3/20 0.34
CYP2C19 P33261 2/20 0.34
ALDH1A1 P00352 3/20 0.33
CACNB4 O00305 2/20 0.33
CACNA1A O00555 2/20 0.33
CACNA1G O43497 2/20 0.33
CACNG3 O60359 2/20 0.33
CACNA1F O60840 2/20 0.33
CACNA1H O95180 2/20 0.33
ACHE P22303 2/20 0.33
CACNB3 P54284 2/20 0.33
CACNA2D1 P54289 2/20 0.33
CACNG7 P62955 2/20 0.33
CACNA1B Q00975 2/20 0.33
CACNA1D Q01668 2/20 0.33
CACNB1 Q02641 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL662261 0.88 LMNA (0.44) LMNAGAAHTTCYP1A2CYP2C9
SCHEMBL662361 0.85 LMNA (0.44) LMNAGAAHTTCYP1A2CYP2C9
SCHEMBL661613 0.76 CYP1A2 (0.43) LMNAGAAHTTCYP1A2CYP2C9
SCHEMBL662728 0.74 LMNA (0.60) LMNAGAAHTTCYP1A2CYP2C9
SCHEMBL663100 0.74 CYP1A2 (0.43) LMNAGAAHTTCYP1A2CYP2C9
SCHEMBL664476 0.72 CYP1A2 (0.40) LMNAGAAHTTCYP1A2CYP2C9
SCHEMBL12423430 0.72 LMNA (0.32) LMNAGAAHTT
SCHEMBL662235 0.70 CYP1A2 (0.40) LMNAGAAHTTCYP1A2CYP2C9
SCHEMBL12424178 0.70 LMNA (0.32) LMNAGAAHTT
SCHEMBL661677 0.70 LMNA (0.42) LMNAGAAHTTCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2536733-B1 TRICYCLIC PYRIDINE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PREPARATION BOEHRINGER INGELHEIM INT (DE) 2014-11-26 EP disclosed