SCHEMBL16263740

SCHEMBL16263740

Cc1cc(C(N)=O)c(NC(=O)c2ccccc2F)s1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
KDM4E B2RXH2 2/20 0.54
LMNA P02545 2/20 0.54
HPGD P15428 1/20 0.54
NPC1 O15118 4/20 0.52
RAB9A P51151 4/20 0.52
SMN1; SMN2 Q16637 4/20 0.51
GLA P06280 1/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
TDP1 Q9NUW8 1/20 0.49
IKBKB O14920 3/20 0.48
HTT P42858 2/20 0.47
TP53 P04637 1/20 0.47
PKM P14618 1/20 0.47
ALOX15 P16050 1/20 0.47
HSD17B10 Q99714 1/20 0.47
JAK2 O60674 2/20 0.47
JAK3 P52333 1/20 0.47
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7003680 0.84 KDM4E (0.63) ALDH1A1KDM4ELMNAHPGDNPC1
SCHEMBL19494363 0.84 NPC1 (0.52) ALDH1A1KDM4ELMNAHPGDNPC1
SCHEMBL19494506 0.83 NPC1 (0.49) ALDH1A1KDM4ELMNAHPGDNPC1
SCHEMBL16246356 0.82 NPC1 (0.48) ALDH1A1KDM4ELMNAHPGDNPC1
SCHEMBL19494877 0.82 NPC1 (0.50) ALDH1A1KDM4ELMNAHPGDNPC1
SCHEMBL19494348 0.81 NPC1 (0.47) ALDH1A1KDM4ELMNAHPGDNPC1
SCHEMBL6504891 0.81 IKBKB (0.57) ALDH1A1KDM4ELMNAHPGDNPC1
SCHEMBL19494902 0.81 NPC1 (0.49) ALDH1A1KDM4ELMNAHPGDNPC1
SCHEMBL16246366 0.80 LMNA (0.51) ALDH1A1KDM4ELMNAHPGDNPC1
SCHEMBL16246509 0.80 NPC1 (0.47) ALDH1A1KDM4ELMNAHPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014180562-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF CYSTIC FIBROSIS GALAPAGOS NV (BE) 2014-11-13 WO disclosed