SCHEMBL1626468

SCHEMBL1626468

CCOC(=O)C1=C(O)c2cc(Cl)ccc2C(C)(C)C1=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SPR P35270 2/20 0.59
KDM4E B2RXH2 6/20 0.42
ALDH1A1 P00352 5/20 0.42
MAPT P10636 3/20 0.42
HPGD P15428 3/20 0.42
LMNA P02545 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
TNF P01375 1/20 0.42
HSP90AA1 P07900 1/20 0.42
ALOX12 P18054 1/20 0.42
CCR6 P51684 1/20 0.42
RUNX1 Q01196 1/20 0.42
CBFB Q13951 1/20 0.42
HKDC1 Q2TB90 1/20 0.42
NOD2 Q9HC29 1/20 0.42
GPR35 Q9HC97 1/20 0.42
NOD1 Q9Y239 1/20 0.42
ABCC1 P33527 1/20 0.40
GAA P10253 1/20 0.40
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1626913 0.90 SPR (0.52) SPRKDM4EALDH1A1MAPTHPGD
SCHEMBL1626493 0.88 SPR (0.57) SPRKDM4EALDH1A1MAPTHPGD
SCHEMBL1625402 0.87 SPR (0.46) SPRKDM4EALDH1A1MAPTHPGD
SCHEMBL1625493 0.87 SPR (0.56) SPRKDM4EALDH1A1MAPTHPGD
SCHEMBL1624395 0.85 SPR (0.45) SPRKDM4EALDH1A1MAPTHPGD
SCHEMBL1627014 0.85 SPR (0.45) SPRKDM4EALDH1A1MAPTHPGD
SCHEMBL1627138 0.85 SPR (0.55) SPRKDM4EALDH1A1MAPTHPGD
SCHEMBL1625783 0.85 SPR (0.46) SPRKDM4EALDH1A1MAPTHPGD
SCHEMBL1626308 0.83 SPR (0.72) SPRKDM4EALDH1A1MAPTHPGD
SCHEMBL1626619 0.83 SPR (0.72) SPRKDM4EALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7928139-B2 Naphthalenone compounds exhibiting prolyl hydroxylase inhibitory activity, compositions, and uses thereof AMGEN INC. (US) 2011-04-19 US disclosed
US-20100048572-A1 NAPHTHALENONE COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS, AND USES THEREOF AMGEN INC. (US) 2010-02-25 US disclosed
US-7635715-B2 Naphthalenone compounds exhibiting prolyl hydroxylase inhibitory activity, compositions, and uses thereof AMGEN INC. (US) 2009-12-22 US disclosed
US-20090093483-A1 Naphthalenone compounds exhibiting prolyl hydroxylase inhibitory activity, compositions, and uses thereof AMGEN INC. (US) 2009-04-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048572-A1 NAPHTHALENONE COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS, AND USES THEREOF EGLN2, EGLN3, HIF1AN SPR 754/4885KDM4E 977/4885ALDH1A1 128/4885
US-20090093483-A1 Naphthalenone compounds exhibiting prolyl hydroxylase inhibitory activity, compositions, and uses thereof EGLN2, EGLN3, HIF1AN SPR 754/4885KDM4E 977/4885ALDH1A1 128/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.