SCHEMBL16274604

SCHEMBL16274604

CCOC(=O)c1c(O)c2cncnc2n(OCc2ccccc2)c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.48
RECQL P46063 1/20 0.47
ALDH1A1 P00352 7/20 0.47
GAA P10253 3/20 0.44
TSHR P16473 3/20 0.44
MAPK1 P28482 2/20 0.44
HSD17B10 Q99714 2/20 0.44
HPGD P15428 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
LMNA P02545 3/20 0.43
MAPT P10636 2/20 0.42
PKM P14618 1/20 0.42
HTT P42858 2/20 0.41
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM5A P29375 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16274700 0.87 PDE4B (0.48) KDM4EALDH1A1GAATSHRMAPK1
SCHEMBL16274683 0.87 ALDH1A1 (0.44) KDM4EALDH1A1GAATSHRMAPK1
SCHEMBL16274845 0.86 RPS6KB1 (0.39) ALDH1A1TSHRMAPK1HSD17B10LMNA
SCHEMBL16274665 0.86 KDM4E (0.48) KDM4ERECQLALDH1A1GAATSHR
SCHEMBL1522959 0.85 KDM4E (0.53) KDM4ERECQLALDH1A1GAATSHR
SCHEMBL16274812 0.85 MAPT (0.46) KDM4EALDH1A1GAATSHRMAPK1
SCHEMBL16274809 0.85 CYP1A2 (0.42) KDM4EALDH1A1TSHRMAPK1HSD17B10
SCHEMBL3516982 0.85 KDM4E (0.47) KDM4ERECQLALDH1A1GAATSHR
SCHEMBL3514749 0.84 KDM4E (0.47) KDM4ERECQLALDH1A1GAATSHR
SCHEMBL3517692 0.84 KDM4E (0.47) KDM4ERECQLALDH1A1GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2810944-A1 HETEROCYCLIC COMPOUND HAVING ANTI-HIV ACTIVITY Toyama Chemical Co., Ltd. (JP) 2014-12-10 EP disclosed