SCHEMBL16299181

SCHEMBL16299181

CCCn1c(=O)n(C2CC2)c(=O)c2[nH]c(-c3ccc(N(CC4CC4)C(=O)c4ccc(I)nc4)nc3)nc21

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 14/20 0.46
ADORA2A P29274 10/20 0.46
CHRM4 P08173 1/20 0.42
ADORA3 P0DMS8 2/20 0.41
ADORA1 P30542 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1243367 0.91 ADORA2B (0.46) ADORA2BADORA2ACHRM4ADORA3ADORA1
SCHEMBL9885749 0.91 ADORA2B (0.45) ADORA2BADORA2ACHRM4ADORA3ADORA1
SCHEMBL16299180 0.91 ADORA2B (0.47) ADORA2BADORA2AADORA3ADORA1
SCHEMBL1002670 0.91 ADORA2B (0.49) ADORA2BADORA2AADORA3ADORA1
SCHEMBL1243464 0.90 ADORA2B (0.49) ADORA2BADORA2ACHRM4ADORA3ADORA1
SCHEMBL1242614 0.90 ADORA2B (0.46) ADORA2BADORA2ACHRM4ADORA3ADORA1
SCHEMBL1243808 0.89 ADORA2A (0.44) ADORA2BADORA2AADORA3ADORA1
SCHEMBL1002030 0.88 ADORA2B (0.45) ADORA2BADORA2AADORA3ADORA1
SCHEMBL17364389 0.86 ADORA2B (0.53) ADORA2BADORA2AADORA3ADORA1
SCHEMBL1243139 0.83 ADORA2B (0.51) ADORA2BADORA2ACHRM4ADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8193200-B2 administering a substituted 8-(3-pyridyl)-xanthine; ulcerative colitis; Crohn's disease UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2012-06-05 US disclosed