SCHEMBL16315367

SCHEMBL16315367

CCN(CC)C(=O)c1ccc(C2=CC3(CCCN(OCOC(C)(C)C)CC3)Oc3cccc(OCOC)c32)cn1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 20/20 0.48
KCNH2 Q12809 18/20 0.48
CYP2D6 P10635 13/20 0.48
MRGPRX2 Q96LB1 1/20 0.39
OPRM1 P35372 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16359483 0.93 OPRD1 (0.50) OPRD1KCNH2CYP2D6MRGPRX2OPRM1
SCHEMBL471474 0.88 OPRD1 (0.48) OPRD1KCNH2CYP2D6MRGPRX2
SCHEMBL16315264 0.83 OPRD1 (0.51) OPRD1KCNH2CYP2D6OPRM1
SCHEMBL12262199 0.83 OPRD1 (0.48) OPRD1KCNH2CYP2D6MRGPRX2
SCHEMBL471472 0.78 OPRD1 (0.52) OPRD1KCNH2CYP2D6MRGPRX2OPRM1
SCHEMBL10257763 0.76 OPRD1 (0.55) OPRD1KCNH2CYP2D6MRGPRX2OPRM1
SCHEMBL16315260 0.76 OPRD1 (0.43) OPRD1KCNH2CYP2D6OPRM1
SCHEMBL467355 0.76 OPRD1 (0.72) OPRD1KCNH2CYP2D6MRGPRX2OPRM1
SCHEMBL12262138 0.74 OPRD1 (0.65) OPRD1KCNH2CYP2D6OPRM1
SCHEMBL471361 0.74 OPRD1 (0.67) OPRD1KCNH2CYP2D6MRGPRX2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399577-A1 Use of N-containing spirocompounds for the enhancement of cognitive function Adolor Corporation (US) 2011-12-28 EP disclosed
WO-2008033299-A2 USE OF N-CONTAINING SPIROCOMPOUNDS FOR THE ENHANCEMENT OF COGNITIVE FUNCTION ADOLOR CORPORATION (US) 2008-03-20 WO disclosed