SCHEMBL16319222

SCHEMBL16319222

COc1ccc(F)c(-c2ccc(OC)nc2CC(C)(C)C)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 4/20 0.47
PDE2A O00408 8/20 0.45
PDE10A Q9Y233 8/20 0.45
PDE6D O43924 1/20 0.45
PDE6A P16499 1/20 0.45
PDE6G P18545 1/20 0.45
PDE4A P27815 1/20 0.45
PDE6B P35913 1/20 0.45
PDE6C P51160 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
PDE3B Q13370 1/20 0.45
PDE6H Q13956 1/20 0.45
PDE3A Q14432 1/20 0.45
GRK6 P43250 1/20 0.40
KDM1A O60341 1/20 0.38
AMY1A P0DUB6 2/20 0.37
IDH2 P48735 1/20 0.37
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16318899 0.87 FFAR1 (0.48) FFAR1PDE2APDE10APDE6DPDE6A
SCHEMBL16318830 0.85 FFAR1 (0.53) FFAR1PDE2APDE10APDE6DPDE6A
SCHEMBL16319376 0.85 FFAR1 (0.51) FFAR1PDE2APDE10APDE6DPDE6A
SCHEMBL16319059 0.85 FFAR1 (0.51) FFAR1PDE2APDE10APDE6DPDE6A
SCHEMBL16318921 0.84 FFAR1 (0.46) FFAR1PDE2APDE10APDE6DPDE6A
SCHEMBL16318621 0.78 FFAR1 (0.56) FFAR1
SCHEMBL16319094 0.77 PDE2A (0.48) PDE2APDE10APDE6DPDE6APDE6G
SCHEMBL16318636 0.77 FFAR1 (0.53) FFAR1GRK6NPC1RAB9A
SCHEMBL16319307 0.75 FFAR1 (0.51) FFAR1GRK6KDM1AAMY1A
SCHEMBL16319375 0.74 FFAR1 (0.51) FFAR1GRK6KDM1AAMY1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382188-B2 Aromatic ring compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-07-05 US disclosed
EP-2816023-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2014-12-24 EP disclosed