SCHEMBL16319094

SCHEMBL16319094

COc1ccc(F)c(-c2ccc(OC)nc2Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 7/20 0.48
PDE10A Q9Y233 7/20 0.48
PDE6D O43924 1/20 0.48
PDE6A P16499 1/20 0.48
PDE6G P18545 1/20 0.48
PDE4A P27815 1/20 0.48
PDE6B P35913 1/20 0.48
PDE6C P51160 1/20 0.48
PDE4B Q07343 1/20 0.48
PDE4C Q08493 1/20 0.48
PDE4D Q08499 1/20 0.48
PDE3B Q13370 1/20 0.48
PDE6H Q13956 1/20 0.48
PDE3A Q14432 1/20 0.48
AMY1A P0DUB6 2/20 0.44
IDH2 P48735 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CYP17A1 P05093 1/20 0.39
CYP11B1 P15538 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16319299 0.81 ALDH1A1 (0.45) AMY1AIDH2NPC1RAB9ACYP17A1
SCHEMBL16318848 0.78 PTPN1 (0.43) AMY1ANPC1RAB9AGRK6
SCHEMBL16319222 0.77 FFAR1 (0.47) PDE2APDE10APDE6DPDE6APDE6G
SCHEMBL15973333 0.76 PDE2A (0.43) PDE2APDE10APDE6DPDE6APDE6G
SCHEMBL8698362 0.74 MAPT (0.40) PDE2APDE10AAMY1AIDH2NPC1
SCHEMBL17436180 0.69 KDM1A (0.45) AMY1AIDH2NPC1RAB9ACYP17A1
SCHEMBL15972269 0.69 ERN1 (0.47) AMY1ANPC1
SCHEMBL16318931 0.68 NPC1 (0.45) NPC1RAB9AHSP90AA1
SCHEMBL8774927 0.68 ALDH1A1 (0.44) AMY1AIDH2NPC1RAB9AGRK6
SCHEMBL1042563 0.67 MAPT (0.56) AMY1ANPC1RAB9AIDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382188-B2 Aromatic ring compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-07-05 US disclosed
EP-2816023-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2014-12-24 EP disclosed