SCHEMBL16319237

SCHEMBL16319237

NC(=O)c1ccc(Oc2ccc(Cl)c(Cl)c2)c(Cl)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.66
HTR2A P28223 2/20 0.66
KCNH2 Q12809 1/20 0.66
CHEK2 O96017 7/20 0.52
ESRRA P11474 1/20 0.48
KMO O15229 1/20 0.48
BCAT2 O15382 1/20 0.48
PARP15 Q460N3 2/20 0.47
PARP14 Q460N5 2/20 0.47
PARP10 Q53GL7 2/20 0.47
TNKS O95271 1/20 0.47
TNKS2 Q9H2K2 1/20 0.47
PARP2 Q9UGN5 1/20 0.47
SLC6A2 P23975 1/20 0.47
SLC6A3 Q01959 1/20 0.47
F2 P00734 1/20 0.46
F10 P00742 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP3A5 P20815 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16319568 0.87 SLC6A4 (0.65) SLC6A4HTR2AKCNH2CHEK2KMO
SCHEMBL364754 0.85 SLC6A4 (0.64) SLC6A4HTR2AKCNH2CHEK2PARP10
SCHEMBL10252664 0.84 SIRT2 (0.53) SLC6A4HTR2AKCNH2CHEK2ESRRA
SCHEMBL27486876 0.83 PARP10 (0.59) SLC6A4HTR2AKCNH2CHEK2PARP15
SCHEMBL367843 0.81 BCAT2 (0.65) SLC6A4HTR2AKCNH2CHEK2KMO
SCHEMBL28866121 0.81 BCAT2 (0.65) SLC6A4HTR2AKCNH2CHEK2KMO
SCHEMBL3701320 0.81 PARP10 (0.65) SLC6A4HTR2AKCNH2CHEK2ESRRA
SCHEMBL11355202 0.79 SLC6A2 (0.58) SLC6A4PARP15PARP14PARP10TNKS
Hydrochloric Acid SCHEMBL4372370 0.79 BCAT2 (0.62) SLC6A4HTR2AKCNH2CHEK2KMO
SCHEMBL3699757 0.77 CHEK2 (0.59) SLC6A4HTR2AKCNH2CHEK2ESRRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed