SCHEMBL16319275

SCHEMBL16319275

COc1ccc(F)c(-c2ccc(O)cc2-c2nnc(C(C)(C)C)o2)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 2/20 0.43
PIK3CB P42338 2/20 0.43
GUSB P08236 5/20 0.41
ALDH1A1 P00352 5/20 0.38
HPGD P15428 3/20 0.38
HSD17B10 Q99714 3/20 0.38
KDM4E B2RXH2 2/20 0.38
LMNA P02545 1/20 0.37
TNIK Q9UKE5 1/20 0.36
FFAR1 O14842 1/20 0.36
TSHR P16473 2/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PTPN1 P18031 1/20 0.36
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TERT O14746 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16318838 0.87 PIK3CD (0.36) PIK3CDPIK3CBALDH1A1HPGDHSD17B10
SCHEMBL16319268 0.75 GUSB (0.41) GUSBALDH1A1TNIKFFAR1MAPT
SCHEMBL16318931 0.73 NPC1 (0.45) ALDH1A1HSD17B10LMNATNIKTSHR
SCHEMBL16318872 0.70 GUSB (0.41) GUSBTNIKMAPTSMN1; SMN2
SCHEMBL16318965 0.70 PTPN1 (0.41) ALDH1A1HPGDHSD17B10KDM4ETNIK
SCHEMBL16319224 0.70 FFAR1 (0.40) PIK3CDPIK3CBTNIKFFAR1
SCHEMBL16318590 0.69 FFAR1 (0.48) ALDH1A1TNIKFFAR1GAA
SCHEMBL16318775 0.69 FFAR1 (0.43) ALDH1A1TNIKFFAR1GAA
SCHEMBL16318940 0.68 FFAR1 (0.41) TNIKFFAR1
SCHEMBL16318863 0.67 FFAR1 (0.38) ALDH1A1FFAR1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382188-B2 Aromatic ring compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-07-05 US disclosed
EP-2816023-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2014-12-24 EP disclosed