SCHEMBL16319268

SCHEMBL16319268

COc1ccc(F)c(-c2ccc(O)cc2-c2nnc(C(C)(C)C)s2)c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GUSB P08236 3/20 0.41
NPC1 O15118 2/20 0.37
MAPT P10636 2/20 0.37
RAB9A P51151 2/20 0.37
TNIK Q9UKE5 1/20 0.36
FFAR1 O14842 1/20 0.36
POLQ O75417 1/20 0.36
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16318872 0.91 GUSB (0.41) GUSBNPC1MAPTRAB9ATNIK
SCHEMBL16319293 0.87 NPC1 (0.39) NPC1MAPTRAB9AFFAR1POLQ
SCHEMBL16318752 0.76 FFAR1 (0.42) FFAR1
SCHEMBL16319275 0.75 PIK3CD (0.43) GUSBMAPTTNIKFFAR1ALDH1A1
SCHEMBL15081838 0.74 ALDH1A1 (0.40) NPC1MAPTRAB9AALDH1A1
SCHEMBL16318931 0.73 NPC1 (0.45) NPC1MAPTRAB9ATNIKALDH1A1
SCHEMBL16318965 0.70 PTPN1 (0.41) MAPTTNIKFFAR1ALDH1A1GAA
SCHEMBL16318590 0.69 FFAR1 (0.48) TNIKFFAR1ALDH1A1GAA
SCHEMBL16318775 0.69 FFAR1 (0.43) TNIKFFAR1ALDH1A1GAA
SCHEMBL16318940 0.68 FFAR1 (0.41) TNIKFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382188-B2 Aromatic ring compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-07-05 US disclosed
EP-2816023-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2014-12-24 EP disclosed