SCHEMBL16319452

SCHEMBL16319452

CS(=O)(=O)NC(=O)c1cc(F)c(Oc2cc(C(F)(F)F)ccc2Cl)cc1F

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 20/20 0.66
SCN5A Q14524 3/20 0.51
SCN1A P35498 1/20 0.51
SCN4A P35499 1/20 0.51
SCN7A Q01118 1/20 0.51
SCN2A Q99250 1/20 0.51
SCN3A Q9NY46 1/20 0.51
SCN8A Q9UQD0 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16319536 0.87 SCN9A (0.54) SCN9ASCN5ASCN1ASCN4ASCN2A
SCHEMBL16319458 0.87 SCN9A (0.54) SCN9ASCN5ASCN1ASCN4ASCN2A
SCHEMBL679928 0.86 SCN9A (0.71) SCN9ASCN5A
SCHEMBL16319614 0.85 SCN9A (0.70) SCN9ASCN5ASCN1A
SCHEMBL16319835 0.83 SCN9A (0.74) SCN9ASCN5ASCN1ASCN4ASCN2A
SCHEMBL16319537 0.82 SCN9A (0.78) SCN9ASCN5A
SCHEMBL16319313 0.81 SCN9A (0.64) SCN9ASCN5A
SCHEMBL16319664 0.81 SCN9A (0.77) SCN9ASCN5A
SCHEMBL17048520 0.81 SCN9A (0.63) SCN9ASCN5ASCN1A
SCHEMBL16319547 0.80 SCN9A (0.68) SCN9ASCN5ASCN1ASCN4ASCN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed