SCHEMBL16319456

SCHEMBL16319456

COc1cc(Oc2ccc(Cl)cc2OC)ccc1C#N

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AR P10275 11/20 0.60
SLC6A4 P31645 2/20 0.49
ESRRA P11474 2/20 0.47
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
SLC22A12 Q96S37 3/20 0.45
KDM4E B2RXH2 1/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A3 Q01959 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11189002 0.90 AR (0.58) ARSLC6A4POLBGAASLC22A12
SCHEMBL363575 0.88 AR (0.51) ARSLC6A4SLC22A12
SCHEMBL4857820 0.86 AR (0.53) ARSLC6A4KDM4EUSP2ALDH1A1
SCHEMBL15094069 0.82 AR (0.66) ARSLC6A4ESRRAKDM4EALDH1A1
SCHEMBL5341215 0.81 AR (0.46) ARESRRAPOLBGAAKDM4E
SCHEMBL5343220 0.81 ALDH1A1 (0.52) ARESRRAPOLBGAAALDH1A1
SCHEMBL5344036 0.80 SLC6A4 (0.60) SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL5344013 0.80 SLC6A4 (0.61) SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL29615609 0.79 ALDH1A1 (0.61) ARSLC6A4KDM4EUSP2ALDH1A1
SCHEMBL945003 0.79 ALDH1A1 (0.61) ARSLC6A4KDM4EUSP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed