SCHEMBL16319657

SCHEMBL16319657

COc1cc(OC(F)(F)F)ccc1Oc1cc(F)c(C(=O)NS(C)(=O)=O)cc1F

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 16/20 0.58
SCN8A Q9UQD0 1/20 0.46
SCN10A Q9Y5Y9 1/20 0.46
SCN7A Q01118 1/20 0.46
SCN5A Q14524 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16319474 0.96 SCN9A (0.58) SCN9ASCN7ASCN5A
SCHEMBL16319491 0.87 SCN9A (0.68) SCN9ASCN7ASCN5A
SCHEMBL16319458 0.85 SCN9A (0.54) SCN9ASCN8ASCN10ASCN5A
SCHEMBL16319893 0.85 SCN9A (0.58) SCN9ASCN8ASCN10ASCN5A
SCHEMBL16319680 0.84 SCN9A (0.64) SCN9ASCN7ASCN5A
SCHEMBL16319364 0.84 SCN9A (0.57) SCN9A
SCHEMBL16319340 0.84 SCN9A (0.57) SCN9ASCN8ASCN10ASCN5A
SCHEMBL16319754 0.83 SCN9A (0.62) SCN9ASCN8ASCN10ASCN5A
SCHEMBL365684 0.82 SCN10A (0.47) SCN9ASCN8ASCN10A
SCHEMBL680139 0.82 SCN9A (0.61) SCN9ASCN8ASCN10ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed