SCHEMBL16319689

SCHEMBL16319689

N#Cc1cc(F)c(Oc2ccc(Cl)c(C(F)(F)F)c2)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AR P10275 9/20 0.48
PLA2G7 Q13093 8/20 0.45
SCN9A Q15858 2/20 0.42
KDR P35968 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365180 0.82 AR (0.60) ARPLA2G7KDR
SCHEMBL24998871 0.79 PLA2G7 (0.48) PLA2G7SCN9A
SCHEMBL9103130 0.78 PLA2G7 (0.47) PLA2G7SCN9A
SCHEMBL17884205 0.78 PLA2G7 (0.53) PLA2G7SCN9A
SCHEMBL25737338 0.78 PLA2G7 (0.56) PLA2G7
SCHEMBL9901518 0.78 PLA2G7 (0.53) PLA2G7
SCHEMBL9108605 0.78 PLA2G7 (0.45) PLA2G7SCN9A
SCHEMBL29851798 0.78 PLA2G7 (0.47) PLA2G7SCN9A
SCHEMBL365436 0.77 SCN9A (0.47) PLA2G7SCN9A
SCHEMBL16319739 0.77 AR (0.78) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed