SCHEMBL1633786

SCHEMBL1633786

CC(C)n1cc(-c2ccc(Cl)c(Cl)c2)c2ccc(NS(C)(=O)=O)cc21

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 8/20 0.68
NR3C1 P04150 7/20 0.68
NR3C2 P08235 7/20 0.68
AR P10275 6/20 0.66
SCN9A Q15858 3/20 0.48
SCN5A Q14524 2/20 0.48
BRD4 O60885 3/20 0.40
KAT2B Q92831 1/20 0.39
KIF11 P52732 1/20 0.39
ABL1 P00519 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
CYP2C8 P10632 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2B6 P20813 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1630814 0.90 PGR (0.73) PGRNR3C1NR3C2ARSCN9A
SCHEMBL1631048 0.88 PGR (0.74) PGRNR3C1NR3C2ARSCN9A
SCHEMBL1631878 0.88 PGR (0.62) PGRNR3C1NR3C2ARSCN9A
SCHEMBL1629438 0.87 PGR (0.80) PGRNR3C1NR3C2ARSCN9A
SCHEMBL1631079 0.87 PGR (0.62) PGRNR3C1NR3C2ARSCN9A
SCHEMBL1630108 0.87 PGR (0.60) PGRNR3C1NR3C2ARSCN9A
SCHEMBL1630553 0.85 PGR (0.64) PGRNR3C1NR3C2ARSCN9A
SCHEMBL1630731 0.85 PGR (0.72) PGRNR3C1NR3C2ARSCN9A
SCHEMBL1629329 0.84 PGR (0.71) PGRNR3C1NR3C2ARSCN9A
SCHEMBL1630826 0.84 PGR (0.74) PGRNR3C1NR3C2ARSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979314-B1 INDOLE SULFONAMIDE MODULATORS OF PROGESTERONE RECEPTORS LILLY CO ELI (US) 2013-01-09 EP disclosed
US-7932284-B2 Indole sulfonamide modulators of progesterone receptors ELI LILLY AND COMPANY (US) 2011-04-26 US disclosed