SCHEMBL1633859

SCHEMBL1633859

NS(=O)(=O)c1ccc(Nc2ncc3cccc(-n4cccn4)c3n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 4/20 0.49
CDK1 P06493 4/20 0.49
CCNB1 P14635 4/20 0.49
CDK9 P50750 4/20 0.49
CDK7 P50613 2/20 0.49
CCNH P51946 2/20 0.49
PIK3CD O00329 1/20 0.47
AURKA O14965 1/20 0.47
DCLK1 O15075 1/20 0.47
PIK3C2G O75747 1/20 0.47
PIK3CG P48736 1/20 0.47
MAPK7 Q13164 1/20 0.47
LRRK2 Q5S007 1/20 0.47
AURKB Q96GD4 1/20 0.47
IKBKB O14920 4/20 0.46
CDK2 P24941 5/20 0.45
IGF1R P08069 1/20 0.45
STK4 Q13043 5/20 0.44
CCNB2 O95067 2/20 0.44
CCNE2 O96020 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1633147 0.78 CDK1 (0.53) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL1635629 0.77 CDK2 (0.55) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL1632497 0.75 AURKA (0.55) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL1634277 0.75 SYK (0.52) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL1633248 0.74 IKBKB (0.53) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL1631112 0.74 IKBKB (0.59) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL1634272 0.73 CA2 (0.49) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL1632468 0.73 MEN1 (0.55) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL1633718 0.72 CDK2 (0.66) CCNT1CDK1CCNB1CDK9PIK3CD
SCHEMBL1634576 0.72 IKBKB (0.58) CCNT1CDK1CCNB1CDK9CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7932262-B2 Quinazolines for PDK1 inhibition NOVARTIS AG (CH) 2011-04-26 US disclosed